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    DERIVATIVES OF [2-(8,9-DIOXO-2,6-DIAZABICYCLO[5.2.0]NON-1(7)-EN-2-YL)ALKYL]PHOSPHONIC ACID AND METHOD OF MAKING THEM
    2.
    发明申请
    DERIVATIVES OF [2-(8,9-DIOXO-2,6-DIAZABICYCLO[5.2.0]NON-1(7)-EN-2-YL)ALKYL]PHOSPHONIC ACID AND METHOD OF MAKING THEM 审中-公开
    [2-（8,9-二氧代-2,6-二氮杂双环[5.2.0] NON-1（7）-EN-2-YL）烷基]磷酸的衍生物及其制备方法

    公开(公告)号：WO2006041975A1

    公开(公告)日：2006-04-20

    申请号：PCT/US2005/035916

    申请日：2005-10-06

    申请人： WYETH ,  BAUDY, Reinhardt, Richard

    发明人： BAUDY, Reinhardt, Richard

    IPC分类号： C07F9/645 ,  A61K31/675 ,  A61P25/02

    CPC分类号： A61K31/551 ,  C07F9/645

    摘要： Compounds of formula (I) or pharmaceutically acceptable salts thereof are provided (Formula I): wherein: A is alkylenyl of 1 to 4 carbon atoms, or alkenylenyl of 2 to 4 carbon atoms; R 1 and R 2 are, independently, hydrogen or a C 5 to C 7 aryl optionally substituted with 1 to 2 substituents, independently, selected from the group consisting of -C(O)R 3 , halogen, cyano, nitro, hydroxyl, C 1 -C 6 alkyl, and C 1 -C 6 alkoxy, with the proviso that at least one of R 1 , and R 2 is not hydrogen; R 3 is, independently, hydrogen, -OR 4 , alkyl, aryl, or heteroaryl; R 4 is hydrogen, alkyl, aryl, or heteroaryl; R 5 and R 6 are, independently, hydrogen, alkyl, hydroxyl, alkoxy, or C 5 to C 7 aryl; wherein any R 3 to R 6 group having an aryl or heteroaryl moiety can optionally be substituted on the aryl or heteroaryl moiety with 1 to about 5 substituents, independently, selected from the group consisting of halogen, cyano, nitro, hydroxyl, C 1 -C 6 alkyl, and C 1 -C 6 alkoxy. Methods of making these compounds as well as methods using the compounds for treating a variety of conditions are also disclosed.

    摘要翻译： 提供式（I）化合物或其药学上可接受的盐（式I）：其中：A为1至4个碳原子的亚烷基或2至4个碳原子的烯基; [R <子

    HERBICIDAL AZA BISPHOSPHONIC ACID COMPOSITIONS
    8.
    发明申请
    HERBICIDAL AZA BISPHOSPHONIC ACID COMPOSITIONS 审中-公开
    除草AZA二磷酸组合物

    公开(公告)号：WO9510188A3

    公开(公告)日：1995-05-04

    申请号：PCT/GB9402183

    申请日：1994-10-07

    申请人： ZENECA LTD

    发明人： FISHER KARL JOSEPH ,  WOOLARD FRANK XAVIER ,  GERDES JOHN MONTGOMERY

    IPC分类号： A01N57/18 ,  A01N57/24 ,  C07F9/38 ,  C07F9/40 ,  C07F9/553 ,  C07F9/568 ,  C07F9/572 ,  C07F9/58 ,  C07F9/59 ,  C07F9/60 ,  C07F9/6503 ,  C07F9/6506 ,  C07F9/6512 ,  C07F9/6518 ,  C07F9/6533 ,  A01N67/18 ,  C07F9/645

    CPC分类号： C07F9/405 ,  A01N57/18 ,  C07F9/3873 ,  C07F9/5532 ,  C07F9/5683 ,  C07F9/5721 ,  C07F9/5722 ,  C07F9/582 ,  C07F9/588 ,  C07F9/591 ,  C07F9/592 ,  C07F9/60 ,  C07F9/65032 ,  C07F9/65061 ,  C07F9/65062 ,  C07F9/65121 ,  C07F9/65181 ,  C07F9/6533

    摘要： Herbicidal compositions comprising: (A) a compound of formula (I), wherein R is hydrogen, hydroxy, C1-C4 alkoxy, halogen, C1-C4 alkyl, C1-C4 haloalkyl, hydroxy-C1-C4-alkyl, hydroxy-C1-C4-alkoxy or N(R )(R ) wherein R and R are each independently hydrogen or C1-C3 alkyl; R and R are each independently hydrogen; hydrocarbyl; substituted hydrocarbyl; hydrocarbyloxy; substituted hydrocarbyloxy; hydrocarbyl-S(O)m-; or substituted hydrocarbyl-S(O)m-; or R and R together form a 3-6 membered carbocyclic ring, optionally substituted with halogen, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 alkylthio or N(R )(R ) wherein R and R are each independently hydrogen or C1-C12 alkyl; and R and R are each independently hydrogen; hydrocarbyl; substituted hydrocarbyl; hydrocarbyloxy; substituted hydrocarbyloxy; hydrocarbylthio; substituted hydrocarbylthio; pyridyl; substituted pyridyl; or are of the formula N(R )(R ) wherein R and R are independently hydrogen, hydrocarbyl or substituted hydrocarbyl; or R and R together with the nitrogen to which they are bound form an aziridine, piperazine, morpholine, thiomorpholine, thiomorpholine sulfinyl, thiomorpholine sulfonyl, hexamethyleneimine, piperidine, tetrahydropyridine, pyrazole, imidazole, pyrrole, triazole, tetrahydropyrimidine, dihydroimidazole, pyrroline, azetidine, perhydroindole, perhydroquinoline, perhydroisoquinoline or pyrrolidine ring, any of which may be optionally substituted with C1-C12 alkyl, halo, C6-C10 aryl, C6-C10 aryl substituted with halo or C1-C6 alkyl, C7-C16 aralkyl, C7-C16 aralkyl substituted with halo or C1-C6 alkyl, nitro, halo-C1-C10-alkyl, C1-C10 alkoxy, C1-C10 alkylthio, C1-C10 alkylsulfonyl, phenoxy, phenoxy substituted with halo or C1-C6 alkyl, C1-C10 alkenyl or cyano; or R and R together with the nitrogen and carbon atoms to which they are bound form an aziridine, piperazine, morpholine, thiomorpholine, thiomorpholine sulfinyl, thiomorpholine sulfonyl, hexamethyleneimine, piperidine, tetrahydropyridine, pyrazole, imidazole, pyrrole, triazole, tetrahydropyrimidine, dihydroimidazole, pyrroline, azetidine, perhydroindole, perhydroquinoline, perhydroisoquinoline or pyrrolidine ring, any of which may be optionally substituted with C1-C12 alkyl, halo, C6-C10 aryl, C6-C10 aryl substituted with halo or C1-C6 alkyl, C7-C16 aralkyl, C7-C16 aralkyl substituted with halo or C1-C6 alkyl, nitro, halo-C1-C10-alkyl, C1-C10 alkoxy, C1-C10 alkylthio, C1-C10 alkylsulfonyl, phenoxy, phenoxy substituted with halo or C1-C6 alkyl, C1-C10 alkenyl or cyano; and m is 0, 1 or 2; and agrochemically acceptable salts thereof; and (B) an agrochemically acceptable carrier therefor. In other aspects, this invention is directed to a method of controlling the growth of plants comprising applying to the area where control is desired an herbicidally effective amount of a compound of formula (I) above; as well as to certain novel compounds having a structure within the scope of formula (I) above.

    摘要翻译： 除草组合物，其包含：（A）式（I）的化合物，其中R 1是氢，羟基，C 1 -C 4烷氧基，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，羟基-C 1 -C 4烷基， 羟基-C 1 -C 4 - 烷氧基或N（R 6）（R 7）（R 7）其中R 6和R 7各自独立地为氢或C 1 -C 3烷基; R 2和R 3各自独立地为氢; 烃基; 取代烃基; 烃; 取代烃氧基; 烃基-S（O）间; 或取代的烃基-S（O）m - ; 或R 2和R 3一起形成3-6元碳环，任选被卤素，羟基，C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6烷硫基或N（R 8）（ R 9）其中R 8和R 9各自独立地为氢或C 1 -C 12烷基; 和R 4和R 5各自独立地为氢; 烃基; 取代烃基; 烃; 取代烃氧基; 烃硫基; 取代的烃基硫代 吡啶基; 取代的吡啶基; 或具有式N（R 10）（R 11）的化合物，其中R 10和R 11独立地为氢，烃基或取代的烃基; 或R 4和R 5与它们所连接的氮一起形成氮丙啶，哌嗪，吗啉，硫代吗啉，硫代吗啉亚硫酰基，硫代吗啉磺酰，六亚甲基亚胺，哌啶，四氢吡啶，吡唑，咪唑，吡咯，三唑，四氢嘧啶 二氢咪唑，吡咯啉，氮杂环丁烷，全氢吲哚，全氢喹啉，全氢异喹啉或吡咯烷环，其中任何一个可以任选被C 1 -C 12烷基，卤素，C 6 -C 10芳基，被卤素或C 1 -C 6烷基取代的C 6 -C 10芳基， C 1-6芳烷基，被卤素或C 1 -C 6烷基取代的C 7 -C 16芳烷基，硝基，卤代-C 1 -C 10 - 烷基，C 1 -C 10烷氧基，C 1 -C 10烷硫基，C 1 -C 10烷基磺酰基，苯氧基，被卤素或C 1取代的苯氧基 -C 1-6烷基，C 1 -C 10烯基或氰基; 或R 2和R 4与它们所连接的氮和碳原子一起形成氮丙啶，哌嗪，吗啉，硫代吗啉，硫代吗啉亚磺酰基，硫代吗啉磺酰，六亚甲基亚胺，哌啶，四氢吡啶，吡唑，咪唑，吡咯， 三唑，四氢嘧啶，二氢咪唑，吡咯啉，氮杂环丁烷，全氢吲哚，全氢喹啉，全氢异喹啉或吡咯烷环，其中任何一个可以任选被C 1 -C 12烷基，卤素，C 6 -C 10芳基，被卤素或C 1 -C 6取代的C 6 -C 10芳基 烷基，C 7 -C 16芳烷基，被卤素或C 1 -C 6烷基取代的C 7 -C 16芳烷基，硝基，卤代-C 1 -C 10 - 烷基，C 1 -C 10烷氧基，C 1 -C 10烷硫基，C 1 -C 10烷基磺酰基，苯氧基， 卤素或C 1 -C 6烷基，C 1 -C 10烯基或氰基; m为0,1或2; 及其农业化学上可接受的盐; 和（B）农业化学上可接受的载体。 在其它方面，本发明涉及一种控制植物生长的方法，其包括向需要控制的区域施用除草有效量的上述式（I）化合物; 以及某些具有上述式（I）范围内的结构的新化合物。

    ２，３－ビスホスフィノピラジン誘導体の製造方法及びホスフィン遷移金属錯体の製造方法
    9.
    发明申请
    ２，３－ビスホスフィノピラジン誘導体の製造方法及びホスフィン遷移金属錯体の製造方法 审中-公开

    公开(公告)号：WO2019031232A1

    公开(公告)日：2019-02-14

    申请号：PCT/JP2018/027702

    申请日：2018-07-24

    申请人： 日本化学工業株式会社

    发明人： 今本　恒雄

    IPC分类号： C07F9/645 ,  C07F1/12 ,  C07F9/50

    摘要： 下記一般式（１）：で表される２，３－ジハロゲノピラジンと、下記一般式（２）：で表される水素－ホスフィンボラン化合物と、脱ボラン化剤と、を含む液に、塩基を添加して反応を行い、下記一般式（３）：で表される２，３－ビスホスフィノピラジン誘導体を得る第一工程を、有することを特徴とする２，３－ビスホスフィノピラジン誘導体の製造方法。本発明によれば、工業的に有利な２，３－ビスホスフィノピラジン誘導体の製造方法を提供することができる。